Melao-motheo ea Nucleic Acid Synthesis

Nucleic acid synthesis e etsoa ho sebelisoa mokhoa o tiileng oa sialic amide triglyceride, moo karolo ea 3' ea DNA e sa sebetseng holim'a karolo e tiileng ea karoloana 'me li-nucleotide li kenngoa ka tsela ea 3' ho ea ho 5' ho fihlela karolo e lakatsehang ea DNA e kopantsoe. .Sena se fapane le tlhahiso ea DNA ka tšebeliso ea DNA polymerase.

Qetello ea 3 ea setsi sa pele ha e sebetse ho CPG nakong ea ho qaptjoa, 5'-OH ea setsi se latelang se sirelelitsoe ka di-p-tolyl trityl DMT, sehlopha sa amino se motheong se sirelelitsoe ka benzoic acid le 3′. -OH e ntan'o sebelisoa ka motsoako oa amino phosphate.Motheo o le mong oa 5 5'-OH oa motheo oa 1 le 3'-OH oa motheo o latelang o etsa phosphite triglyceride, eo ka nako eo e nang le oxidized ka iodine ho phosphate triglyceride, mosireletsi motheong oa bobeli 5'-OH o tlosoa ke ho eketsa dichloroacetic acid DM cycles ka ho eketsoa ha setsi se latelang, 'me ka mor'a ho kopanya mosireletsi ho 5'-OH o tlosoa ka acid e fokolang Sekhechana se khaotsoe ho tloha ho resin e tiileng ka concentrated ammonium hydroxide, mosireletsi o tlosoa motheong. ka concentrated ammonium hydroxide tlas'a ho futhumala, ammonium hydroxide e tlosoa, sekhechana se omisitsoe, 'me nucleic acid e hloekisoa ke liquid chromatography kapa PAGE.

 

Mehato ea Oligo Synthesis

Deblocking

TheSehlopha sa 5 se sireletsang DMT se tlosoa ka ho eketsa tharollo ea TCA.

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Tshebetso

Ho kopanya activator le oligonucleotide monomer ho theha oligonucleotide monomer e sebetsang lipakeng.

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Ho kopanya

Sehlopha sa 5-terminal hydroxyl se sebetsana le oligonucleotide e sebetsang ka hare ho anti-generative condensation reaction ho theha bond e sa tsitsang ea phosphite triglyceride.

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Capping 

Ho eketsoa ha capping agent ho etsa acetylation capping reaction ka lihlopha tse feteletseng tsa hydroxyl tse sa ameheng karabelong ea condensation.

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Oxidation 

Ho eketsoa ha tharollo ea iodine e nang le metsi e sebetsana le litlamo tse sa tsitsang tsa phosphite ka oxidation ho theha maqhama a tsitsitseng a phosphoric acid triglyceride.

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Cyanoethyl Cleavage

Sehlahisoa sa nucleic acid ka mor'a ho kopanya, ka ho eketsoa ha tharollo ea DEA ho tlosa sehlopha sa cyanoethyl ho tloha ho phosphate triglyceride bond.

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Khiloe & Tšireletso

Likaroloana tsa asiti ea nucleic li petsoha ho sejari sa mohato o tiileng ka ho eketsa tharollo ea ammonium hydroxide e tebileng ebe e futhumatsoa ho tlosa lihlopha tse sirelletsang litlamong tsa hydrogen tsa metheo.

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Nako ea poso: Nov-21-2022